Biological Activity
Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin release in the rat nucleus accumbens.Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Additional Information
Background References
-
Structural basis for the binding specificity of a SSTR1-selective analog of somatostatin.
Chen et al.
Biochem.Biophys.Res.Commun., 1999;258:689 -
Potent somatostatin undecapeptide agonists selective for somatostatin receptor 1 (sst1).
Rivier et al.
J.Med.Chem., 2001;44:2238 -
The somatostatin receptor (sst1) modulates the release of somatostatin in the nucleus accumbens of the rat.
Vasilaki et al.
Neuropharmacology, 2004;47:612
Product Datasheets
Reconstitution Calculator
Molarity Calculator
FAQs
No product specific FAQs exist for this product, however you may
View all Peptide FAQsVersaClone cDNA Plasmids
Reviews for CH 275
There are currently no reviews for this product. Be the first to review CH 275 and earn rewards!
Have you used CH 275?
Submit a review and receive an Amazon gift card.
$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image