High affinity adenosine A3
receptor antagonist (Ki
= 47 nM) that displays > 200-fold selectivity versus A1
Soluble to 50 mM in DMSO
Desiccate at RT
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
"Reversine" and its 2-substituted adenine derivatives as potent and selective A3 adenosine receptor antagonists.
Perreira et al.
Adenosine receptors as therapeutic targets.
Jacobson and Gao
Nat.Rev.Drug Discov., 2006;5:247
Progress in the pursuit of therapeutic adenosine receptor antagonists.
Moro et al.
The citations listed below are publications that use Tocris products. Selected citations for MRS 3777 hemioxalate include:
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