Biological Activity High affinity D4 receptor ligand; selective over D1, D2, D3 and D5 receptors. Displays antagonist activity at the human D4.2 receptor (Ki = 3.6 nM in transfected CHO cells) and exhibits agonist activity at the D4.4 receptor in HEK 293 cells.
Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
Store at +4°C
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For batch specific data refer to the Certificate of Analysis.
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