Catalog Number: 4919
Biological Activity
Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.
Technical Data
  • M.Wt:
    1008.19
  • Formula:
    C51H69N13O9
  • Sequence:
    XDXXRWK

    (Modifications: X-1 = Ac-Nle, X-3 = beta-Ala, X-4 = D-2-Nal, Lys-7 = C-terminal amide, Asp-2, Lys-7, Cyclized)

  • Solubility:
    Soluble to 1 mg/ml in 25% ethanol / water
  • Storage:
    Store at -20°C
  • CAS No:
    944111-22-2
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: their activity and selectivity at human melanocortin receptors 3, 4, and 5.
    Grieco et al.
    Peptides., 2007;28:1191

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