Histamine H1 Receptor Antagonists: Products

Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines. It has been detected as a mixture of monomers and homodimers, with highest concentration in the placenta, followed by brain, lung (produced by airway smooth muscle, bronchial epithelium and macrophages) and other tissues.

Showing 1-18 out of 18 Histamine H1 Receptor Antagonists Products

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Doxepin hydrochloride


Highly potent H1 antagonist. Also binds to H4 receptor
0508 
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Mirtazapine


Potent 5-HT2 antagonist. Also 5-HT3, H1 and alpha2-antagonist. Antidepressant
20182  
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Astemizole


Orally active, potent H1 antagonist. Also KV11.1 (hERG) channel blocker.
34891  
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Clemizole hydrochloride


TRPC5 blocker; also H1 antagonist
5371 
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Terfenadine


H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker
39482  
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(S)-(+)-Dimethindene maleate


M2-selective antagonist
1425 
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Clemastine fumarate


H1 antagonist
14531  
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Ketotifen fumarate


H1 antagonist
0784 
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Cetirizine dihydrochloride


Selective H1 antagonist
25773  
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trans-Triprolidine hydrochloride


Standard H1 antagonist, highly potent
06622  
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Zotepine


5-HT2A/D2 antagonist; atypical antipsychotic
3996 
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Olopatadine hydrochloride


H1 antagonist; ocular antiallergic agent
4241 
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Diphenhydramine hydrochloride


H1 receptor antagonist
3072 
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Mepyramine maleate


Selective H1 inverse agonist
06601  
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Meclizine dihydrochloride


Human pregnane X receptor agonist; H1 antagonist
4245 
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Loratidine


Peripheral H1 antagonist; antiallergic agent
1944 
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Fexofenadine hydrochloride


H1 receptor antagonist; non-sedating antiallergic agent
24291  
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Desloratadine


High affinity H1 antagonist; anti-inflammatory.
5958 
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