Nicotinic Acetylcholine R alpha 4/CHRNA4: Products

CHRNA4 is a nicotinic acetylcholine receptor, which belongs to a superfamily of ligand-gated ion channels that play a role in fast signal transmission at synapses. These pentameric receptors can bind acetylcholine, which causes an extensive change in conformation that leads to the opening of an ion-conducting channel across the plasma membrane. CHRNA4 is an integral membrane receptor subunit that can interact with either nAChR beta-2 or nAChR beta-4 to form a functional receptor. Mutations in CHRNA4 cause nocturnal frontal lobe epilepsy type 1. Polymorphisms in CHRNA4 that provide protection against nicotine addiction have been described.

Showing 1-18 out of 18 Nicotinic Acetylcholine R alpha 4/CHRNA4 Products

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Dihydro-β-erythroidine hydrobromide


Antagonist for neuronal α4-containing nicotinic receptors
234919  
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A 85380 dihydrochloride


High affinity and selective α4β2 agonist
5017 
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ABT 089 dihydrochloride


High affinity and selective α4β2 partial agonist
5079 
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TC 2559 difumarate


Selective partial agonist at α4β2 receptors
27371  
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Varenicline tartrate


Orally active, subtype-selective α4β2 partial agonist
37542  
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CC4


High affinity and subtype-selective α6β2 and α4β2 partial agonist
5236 
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RJR 2403 oxalate


α4β2 selective nicotinic agonist
10536  
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DMAB-anabaseine dihydrochloride


Partial agonist at α7 nAChR; also α4β2 antagonist
2241 
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3-Bromocytisine


Potent agonist of α4β4, α4β2 and α7 nACh receptors
35491  
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SIB 1508Y maleate


Potent agonist of α4β2, α2β4, α4β4 and α3β4 nACh receptors
4766 
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5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative


Precursor to 5-Iodo-A-85380 (Cat. No. 1518)
1527 
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3-pyr-Cytisine


High affinity, partial agonist of α4β2 receptors
4125 
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Desformylflustrabromine hydrochloride


Positive allosteric modulator of α4β2; also muscle-type nAChR inhibitor
3328 
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5-Iodo-A-85380 dihydrochloride


High affinity α4β2 and α6β2 subtype-selective agonist
15183  
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NS 9283


Positive allosteric modulator of α4β2
5112 
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UB 165 fumarate


Subunit selective nAChR agonist
1348 
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Sazetidine A dihydrochloride


α4β2 receptor ligand; may act as an agonist or a desensitizer
27362  
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Human nAChR alpha 4/CHRNA4 (NP_000735) VersaClone cDNA

RDC0281 
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