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Wnt/β-catenin signaling inhibitor; axin stabilizer
Inhibitor of Hedgehog (Hh) signaling
GLI antagonist; inhibits Hedgehog (Hh) signaling
Selective Hsp90 inhibitor
ARFGAP1 inhibitor; modulates Wnt/β-catenin signaling
STAT3 inhibitor; also inhibits mTORC1 signaling
Breast cancer stem cell inhibitor
Inhibits SUMOylation by binding E1
Selectively kills mutant HRAS-expressing cells; glutathione peroxidase inhibitor; induces ferroptosis
ALDH1A inhibitor; depletes CD133+ cancer stem cells
ALDH1A inhibitor; depletes CD133+ cancer stem cells (CSC)
Potent CXCR1 and CXCR2 allosteric antagonist