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Non-competitive NMDA antagonist; acts at ion channel site
Broad spectrum glutamatergic antagonist
GluN2B-selective NMDA antagonist
Potent NMDA antagonist; acts at glycine site
Highly potent NMDA antagonist
Specific σ ligand, NMDA antagonist
NMDA antagonist; acts at glycine site
Competitive NMDA antagonist
Potent and selective NMDA antagonist; acts at the glycine site
Potent and noncompetitive NMDA antagonist
NMDA antagonist; antidepressant; may not display psychotomimetic or addictive side effects of (S)-ketamine