7 results for "glucagon-receptor-antagonists&view=expanded" in Products

Potent, orally active human glucagon receptor antagonist

Chemical Name: 4-[3-(5-Bromo-2-propoxyphenyl)-5-(4-chlorophenyl)-1H-pyrrol-2-yl]pyridine
Purity: ≥98%
Potent, orally active human glucagon receptor antagonist
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Potent GLP-1 receptor antagonist

Purity: ≥95%
Potent GLP-1 receptor antagonist
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Glucagon receptor antagonist

Purity: ≥95%
Glucagon receptor antagonist
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Peptide antagonist of glucagon-like peptide-2 (GLP-2) receptor

Purity: ≥90%
Peptide antagonist of glucagon-like peptide-2 (GLP-2) receptor
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Negative allosteric modulator of glucagon and GLP-1 receptors

Chemical Name: 4-[[(4-Cyclohexylphenyl)[[[3-(methylsulfonyl)phenyl]amino]carbonyl]amino]methyl]-N-2H-tetrazol-5-ylbenzamide
Purity: ≥98%
Negative allosteric modulator of glucagon and GLP-1 receptors
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Metabolite of GLP-1-(7-36) (Cat. No. 2082)

Alternate Names: Glucagon-like peptide 1 (9-36) amide
Purity: ≥95%
Metabolite of GLP-1-(7-36) (Cat. No. 2082)
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Non-competitive GLP-1 antagonist; orally bioavailable and brain penetrant

Chemical Name: 7-(4-Chlorophenyl)-5,8-dihydro-1,3-dimethyl-5,5-bis(trifluoromethyl)pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione
Purity: ≥98%
Non-competitive GLP-1 antagonist; orally bioavailable and brain penetrant
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