8 results for "mas-related-g-protein-coupled-receptor-agonists&view=expanded" in Products

Endogenous neuropeptide; binds sst1 - sst5, ghrelin receptor and MRGPRX2

Alternate Names: CST-14
Purity: ≥95%
Endogenous neuropeptide; binds sst1 - sst5, ghrelin receptor and MRGPRX2
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Potent MRGPRX1 agonist

Purity: ≥95%
Potent MRGPRX1 agonist
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MRGPRX2 agonist; also non-competitive nAChR antagonist

Purity: ≥95%
MRGPRX2 agonist; also non-competitive nAChR antagonist
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Potent MRGPRX2 agonist

Purity: ≥95%
Potent MRGPRX2 agonist
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MRGPRX2 agonist

Chemical Name: (3R)-N,N-Dimethyl-1-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)-3-pyrrolidinamine
Purity: ≥98%
MRGPRX2 agonist
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Potent C5a receptor antagonist

Purity: ≥95%
Potent C5a receptor antagonist
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Endogenous NPFF1 and NPFF2 agonist; also MRGPRA agonist

Purity: ≥95%
Endogenous NPFF1 and NPFF2 agonist; also MRGPRA agonist
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Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels

Alternate Names: A-4166,Senaglinide
Chemical Name: N-[[4-(1-Methylethyl)cyclohexyl]carbonyl]-D-phenylalanine
Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels
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