6 results for "nrf2-inhibitors&view=expanded" in Products

Nrf2 inhibitor; phenotypically lethal

Chemical Name: N-[4-[2,3-Dihydro-1-(2-methylbenzoyl)-1H-indol-5-yl]-5-methyl-2-thiazolyl]-1,3-benzodioxole-5-acetamide
Purity: ≥98%
Nrf2 inhibitor; phenotypically lethal
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PGK1 inhibitor; activates Nrf2

Chemical Name: (3R,4S)-rel-4-[(4-Chlorophenyl)sulfonyl]tetrahydro-N-(2-methylpropyl)-3-thiophenamine-1,1-dioxide
Purity: ≥98%
PGK1 inhibitor; activates Nrf2
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Caspase-1 and NLRP3 inflammasome inhibitor

Chemical Name: Ethyl 2[(2-chlorophenyl)(hydroxy)methyl]acrylate
Purity: ≥98%
Caspase-1 and NLRP3 inflammasome inhibitor
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Nrf2 activator; inhibits Nrf2/Keap1 interaction

Chemical Name: (3S)-1-[4-[[(2,3,5,6-Tetramethylphenyl)sulfonyl]amino]-1-naphthalenyl]-3-pyrrolidinecarboxylic acid
Purity: ≥98%
Nrf2 activator; inhibits Nrf2/Keap1 interaction
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Inhibitor of Keap1- Nrf2 interaction

Alternate Names: LH601A
Chemical Name: (1S,2R)-2-[[(1S)-1-[(1,3-Dihydro-1,3-dioxo-2H-isoindol-2-yl)methyl]-3,4-dihydro-2(1H)-isoquinolinyl]carbonyl]cyclohexanecarboxylic acid
Purity: ≥98%
Inhibitor of Keap1- Nrf2 interaction
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Covalent allosteric NRF2 inhibitor

Chemical Name: 1-[(3R)-3-[3-(4-Amino-1,3,5-triazin-2-yl)-5-chlorophenyl]-4-morpholinyl]-2-propen-1-one
Purity: ≥98%
Covalent allosteric NRF2 inhibitor
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