17 results for "trpv-antagonists&view=expanded" in Products

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Capsazepine

Catalog #: 0464
Citations (247)
Product Documents

TRPV antagonist; also activator of ENaCδ

Chemical Name: N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide
Purity: ≥98%
TRPV antagonist; also activator of ENaCδ

AMG 9810

Catalog #: 2316
(1)
Citations (92)
Product Documents

Potent and selective TRPV1 competitive antagonist

Chemical Name: (2E)-N-(2,3-Dihydro-1,4-benzodioxin-6-yl)-3-[4-(1,1-dimethylethyl)phenyl]-2-propenamide
Purity: ≥98%
Potent and selective TRPV1 competitive antagonist

SB 366791

Catalog #: 1615
Citations (92)
Product Documents

Potent and selective TRPV1 competitive antagonist

Chemical Name: 4'-Chloro-3-methoxycinnamanilide
Purity: ≥98%
Potent and selective TRPV1 competitive antagonist

A 784168

Catalog #: 4319
Citations (13)
Product Documents

Potent and selective TRPV1 antagonist

Chemical Name: 3,6-Dihydro-3'-(trifluoromethyl)-N-[4-[(trifluoromethyl)sulfonyl]phenyl]-[1(2H),2'-bipyridine]-4-carboxamide
Purity: ≥98%
Potent and selective TRPV1 antagonist

HC 067047

Catalog #: 4100
(2)
Citations (98)
Product Documents

Potent and selective TRPV4 antagonist

Chemical Name: 2-Methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide
Purity: ≥98%
Potent and selective TRPV4 antagonist

GSK 2193874

Catalog #: 5106
Citations (40)
Product Documents

Potent and selective TRPV4 antagonist; orally active

Chemical Name: 3-([1,4'-Bipiperidin]-1'-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2-[3-(trifluoromethyl)phenyl]-4-quinolinecarboxamide
Purity: ≥98%
Potent and selective TRPV4 antagonist; orally active

SET 2

Catalog #: 6990
Citations (7)
Product Documents

Selective TRPV2 antagonist

Chemical Name: N-(2-Furanylmethyl)-3-[[4-(methylpropylamino)-6-(trifluoromethyl)-2-pyrimidinyl]thio]propanamide
Purity: ≥98%
Selective TRPV2 antagonist

JNJ 17203212

Catalog #: 3361
Citations (14)
Product Documents

Reversible, competitive and potent TRPV1 antagonist

Chemical Name: 4-[3-(Trifluoromethyl)-2-pyridinyl]-N-[5-(trifluoromethyl)-2-pyridinyl]-1-piperazinecarboxamide
Purity: ≥98%
Reversible, competitive and potent TRPV1 antagonist

RN 1734

Catalog #: 3746
Citations (45)
Product Documents

Selective TRPV4 antagonist

Chemical Name: 2,4-Dichloro-N-isopropyl-N-(2-isopropylaminoethyl)benzenesulfonamide
Selective TRPV4 antagonist

TRPV3 74a

Catalog #: 6831
Citations (1)
Product Documents

Selective TRPV3 antagonist; brain penetrant

Chemical Name: (αS)-α-[cis-3-Hydroxy-3-methyl-1-[4-(trifluoromethyl)-2-pyridinyl]cyclobutyl]-2-pyridinemethanol
Purity: ≥98%
Selective TRPV3 antagonist; brain penetrant
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