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ARN 272

Catalog #: 4574 Datasheet / COA / SDS

Discontinued Product

4574 has been discontinued.
View all Fatty Acid Amide Hydrolase (FAAH) Inhibitors products.
ARN 272 | CAS No. 488793-85-7 | Fatty Acid Amide Hydrolase (FAAH) Inhibitors
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Description: FAAH-like anandamide transporter (FLAT) inhibitor

Chemical Name: 4-[[4-(4-Hydroxyphenyl)-1-phthalazinyl]amino]-N-phenylbenzamide

Purity: ≥98%

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Biological Activity

FAAH-like anandamide transporter (FLAT) inhibitor (IC50 = 1.8 μM); cytosolic variant of FAAH-1 that binds anandamide. Attenuates anandamide internalization and deactivation in vitro and in vivo respectively. Exhibits analgesic effects in rodent models of CB1-mediated nociceptive and inflammatory pain.

Technical Data

M.Wt:
432.47
Formula:
C27H20N4O2
Solubility:
Soluble to 100 mM in DMSO and to 20 mM in ethanol
Purity:
≥98%
Storage:
Store at RT
CAS No:
488793-85-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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