BML-190
Discontinued Product
Chemical Name: 1-(4-Chlorobenzoyl)-5-methoxy-2-methyl-1-[2-(4-morpholinyl)-2-oxoethyl]-1H-indole
Purity: ≥99%
Biological Activity
Potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively).Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
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Suppression of nerve growth factor Trk receptors and prolactin receptors by endocannabinoids leads to inhibition of human breast and prostate cancer cell proliferation.
Melck et al.
Endocrinology, 2000;141:118 -
New class of potent ligands for the human peripheral cannabinoid receptor.
Gallant et al.
Bioorg.Med.Chem.Lett., 1996;6:2263
Product Datasheets
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Citation for BML-190
The citations listed below are publications that use Tocris products. Selected citations for BML-190 include:
1 Citation: Showing 1 - 1
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In vitro metabolism of indomet. morpholinylamide (BML-190), an inverse agonist for the peripheral cannabinoid receptor (CB(2)) in rat liver microsomes.
Authors: Zhang Et al.
Eur J Pharm Sci 2010;41:163
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