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L803

Catalog #: 2235 Datasheet / COA / SDS

Discontinued Product

2235 has been discontinued.
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L803
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Description: Substrate-competitive inhibitor of GSK-3
Product Details
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Biological Activity Technical Data Additional Information Background Product Datasheets Calculators

Biological Activity

Novel phosphopeptide derived from GSK-3 recognition motif that acts as a substrate-competitive inhibitor of GSK-3β (IC50 = 150 μM). Displays minimal inhibition of Cdc2, MAPK, PKA, CK2, PKCδ and PKB at 200 μM.

Technical Data

M.Wt:
1198.23
Formula:
C50H80N13O19P
Sequence:
KEAPPAPPQSP

(Modifications: Ser-10 = pSer)

Solubility:
Soluble to 1 mg/ml in water
Storage:
Desiccate at -20°C
CAS No:
348089-28-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under licence from Tel Aviv University Future Technology LP

Background References

  1. Ins mimetic action of synthetic phosphorylated peptide inhibitors of glycogen synthase kinase-3.
    Plotkin et al.
    J.Pharmacol.Exp.Ther., 2003;305:974

Product Datasheets

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Reconstitution Calculator

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