CGP 13501

Key Product Details

Product Description

CGP 13501 is a positive allosteric modulator of GABA_B receptors, potentiating the effects of GABA at this receptor type.

Product Specifications for CGP 13501

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for CGP 13501

The following data is based on the product molecular weight 290.44.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	3.44 mL	17.22 mL	34.43 mL
5 mM	0.69 mL	3.44 mL	6.89 mL
10 mM	0.34 mL	1.72 mL	3.44 mL
50 mM	0.07 mL	0.34 mL	0.69 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Urwyler Positive allosteric modulation of native and recombinant γ-aminobutyric acid_B receptors by 2,6-di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its aldehyde analog CGP13501. Mol.Pharmacol. 2001 PMID: 11641424

Product Documents for CGP 13501