Chemical Name: 2-Chloro-N-cyclopentyl-2'-methyladenosine
Biological Activity Potent and highly selective agonist at A1 adenosine receptors (Ki values are 3.3, 9580, 37600 and 1150 nM for human recombinant A1, A2A, A2B and A3 receptors respectively). Acts as a full agonist; inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC50 value of 13.1 nM.
Soluble to 25 mM in DMSO
Store at +4°C
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