CID 2011756

Key Product Details

Product Description

CID 2011756 is a protein kinase D (PKD) inhibitor (IC₅₀ values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively). Cell permeable (EC₅₀ = 10 μM for PKD1 inhibition). ATP-competitive.

Product Specifications for CID 2011756

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for CID 2011756

The following data is based on the product molecular weight 396.87.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

1 Recalculate

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.5 mM	5.04 mL	25.20 mL	50.39 mL
2.5 mM	1.01 mL	5.04 mL	10.08 mL
5 mM	0.50 mL	2.52 mL	5.04 mL
25 mM	0.10 mL	0.50 mL	1.01 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Sharlow Discovery of diverse small molecule chemotypes with cell-based PKD1 inhibitory activity. PLoS One 2011 PMID: 21998636

Product Documents for CID 2011756