Cinanserin hydrochloride

Key Product Details

Product Description

Cinanserin hydrochloride is a 5-HT₂ antagonist. Also inhibits 3C-like proteinase (3CL^pro; M^pro). Inhibits replication of SARS-CoV.

Product Specifications for Cinanserin hydrochloride

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for Cinanserin hydrochloride

The following data is based on the product molecular weight 376.94.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.5 mM	5.31 mL	26.53 mL	53.06 mL
2.5 mM	1.06 mL	5.31 mL	10.61 mL
5 mM	0.53 mL	2.65 mL	5.31 mL
25 mM	0.11 mL	0.53 mL	1.06 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 13 publications citing the usage of this product.

• Pierce Molecular structure basis of ligand selectivity for 5-HT₂ versus 5-HT_1C cortical receptors. Naunyn Schmiedebergs Arch.Pharmacol. 1992 PMID: 1407003
• Chen Cinanserin is an inhibitor of the 3C-like proteinase of the severe acute respiratory syndrome coronavirus and strongly reduces virus replication in vitro. J.Virol. 2005 PMID: 15890949
• Leysen Receptor binding profile of R-41-468, a novel antagonist at 5HT₂ receptors. Life Sci. 1981 PMID: 6261070

Product Documents for Cinanserin hydrochloride