Non-steroidal selective estrogen receptor modulator (SERM). Displays higher affinity for estrogen receptor β
) than for ERα
Soluble to 10 mM in DMSO
Store at +4°C
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Characterization of the pharmacore properties of novel selective estrogen receptor downregulators (SERDs).
Kieser et al.
Fluorine-substituted cyclofenil derivatives as estrogen receptor ligands: synthesis and structure-affinity relationship study of potential PET agents for imaging estrogen receptors in breast cancer.
Seo et al.