FR 139317

Catalog # Availability Size / Price Qty
1210/10
1210/50
FR 139317 | CAS No. 142375-60-8 | Endothelin ETA Receptor Antagonists
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Description: Highly potent, selective ETA antagonist

Chemical Name: N-[N-[N-[(Hexahydro-1H-azepin-1-yl)carbonyl]-L-leucyl]-1-methyl-D-tryptophyl]-3-(2-pyridinyl)-D-alanine

Purity: ≥99%

Product Details
Citations (1)
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Biological Activity

FR 139317 is a highly potent and selective ETA endothelin receptor antagonist (Ki values are 1 nM and 7.3 μM at ETA and ETB subtypes respectively). Active in vivo.

Technical Data

M.Wt:
604.75
Formula:
C33H44N6O5
Solubility:
Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
Purity:
≥99%
Storage:
Desiccate at +4°C
CAS No:
142375-60-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citation for FR 139317

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