Endogenous potent and highly selective bradykinin B1
receptor agonist (Ki
values are 0.12 and > 30000 nM at human B1
receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo
. 16-fold more potent than [Des-Arg9]-Bradykinin
(Cat No. 3005).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Classification of kinin receptors.
Regoli et al.
Hypotensive effects of Lys-des-Arg9-Bradykinin and metabolically protected agonists of B1 receptors for kinins.
Drapeau et al.
International union of pharmacology. LV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences.
Leeb-Lundberg et al.