SB 243213 dihydrochloride

Catalog # Availability Size / Price Qty
3527/10
3527/50
5-HT2C Receptor Inverse Agonists Small Molecule
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Description: Selective 5-HT2C inverse agonist

Chemical Name: 2,3-Dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-6-(trifluoromethyl)-1H-Indole-1-carboxamide dihydrochloride

Purity: ≥99%

Product Details
Citations (1)
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Biological Activity

Selective 5-HT2C inverse agonist (pKb = 9.8). Displays selectivity over other 5-HT2 subtypes (pKi values are 6.8, 7.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C respectively); also exhibits >100-fold selectivity over 50 other receptors, ion channels and enzymes. Displays anxiolytic activity in rat models.

Technical Data

M.Wt:
501.33
Formula:
C22H19F3N4O2.2HCl
Solubility:
Soluble to 50 mM in DMSO
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
1780372-25-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citation for SB 243213 dihydrochloride

The citations listed below are publications that use Tocris products. Selected citations for SB 243213 dihydrochloride include:

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