Peptide agonist for sst₂ and sst₅ somatostatin receptors. IC₅₀/K_d values (nM) at cloned human somatostatin receptors are: > 1000 (sst₁), 0.2 - 1.5 (sst₂), 27 - 36 (sst₃), > 127 (sst₄), and 0.06 - 23 (sst₅).

Product Specifications for Seglitide

Molecular Weight

808.98

Formula

C₄₄H₅₆N₈O₇

Storage

Desiccate at -20°C

CAS Number

81377-02-8

PubChem ID

5311430

InChI Key

NPJIOCBFOAHEDO-AVWFULIKSA-N

SMILES

CC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)[C@H](C)N(C)C(=O)[C@H](CC2=CC=CC=C2)NC1=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Soluble to 1mg/ml in water

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Background References

References are publications that support the biological activity of the product.

Raynor Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding to linear peptides. Mol.Pharmacol. 1993 PMID: 8100350
Hannon Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci.
Hoyer Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch.Pharmacol. 1994 PMID: 7870182

Product Documents for Seglitide

Certificate of Analysis

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Download SDS

Product Specific Notices for Seglitide

For research use only

Related Research Areas

Metabolic Peptide Hormones and Regulators

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Seglitide

Tocris Bioscience | Catalog # 1836

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Product Description