Biological Activity Potent and selective GluK1 (formally GluR5) containing kainate receptor antagonist (IC50 = 7 nM) that displays selectivity over GluK2 (formally GluR6) containing kainate, NMDA, AMPA and group I mGlu receptors. Reversibly blocks induction of NMDA receptor-independent long term potentiation (LTP) in vitro at nanomolar concentrations.
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