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CP 316819

Catalog #: 3542
2 Citations Datasheet / COA / SDS
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3542/10
3542/50

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CP 316819 | CAS No. 186392-43-8 | Phosphorylase Inhibitors
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Description: Selective glycogen phosphorylase inhibitor

Chemical Name: 5-Chloro-N-[(1S,2R)-2-hydroxy-3-(methoxymethylamino)-3-oxo-1-(phenylmethyl)propyl]-1H-indole-2-carboxamide

Purity: ≥98%

Product Details
Citations (2)
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Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

CP 316819 is a selective glycogen phosphorylase inhibitor [IC50 values are 0.017 and 0.034 μM against human skeletal muscle glycogen phosphorylase a (huSMGPa) and liver glycogen phosphorylase a (huLGPa) respectively]. Antihyperglycemic agent.

Technical Data

M.Wt:
415.87
Formula:
C21H22ClN3O4
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥98%
Storage:
Store at RT
CAS No:
186392-43-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for CP 316819

The citations listed below are publications that use Tocris products. Selected citations for CP 316819 include:

2 Citations: Showing 1 - 2

  1. Glycogen metabolism is dispensable for tumour progression in clear cell renal cell carcinoma.
    Authors: Jun Et al.
    Nat Metab  2021;3:327-336
  2. Energy substrates that fuel fast neuronal network oscillations.
    Authors: Galow Et al.
    J Exp Bot  2014;8:398

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