Cyanopindolol hemifumarate

Key Product Details

Product Description

Cyanopindolol hemifumarate is a 5-HT_1A/1B antagonist with roughly equal affinity at each receptor; also a β-adrenoceptor antagonist.

Product Specifications for Cyanopindolol hemifumarate

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for Cyanopindolol hemifumarate

The following data is based on the product molecular weight 345.40.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	2.90 mL	14.48 mL	28.95 mL
5 mM	0.58 mL	2.90 mL	5.79 mL
10 mM	0.29 mL	1.45 mL	2.90 mL
50 mM	0.06 mL	0.29 mL	0.58 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 12 publications citing the usage of this product.

• Blue Interaction of dihydroalprenolol and cyanopindolol with atypical β-adrenoceptors in guinea-pig ileum. Br.J.Pharmacol.
• Giles Characterization of a 5-HT_1B receptor on CHO cells: functional responses in the absence of radioligand binding. Br.J.Pharmacol. 1996 PMID: 8882605
• Hoey Atypical responses of rat ileum to pindolol, cyanopindolol and iodocyanopindolol. Br.J.Pharmacol. 1996 PMID: 8646418
• Engel Identity of presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1_B binding sites. Naunyn Schmiedebergs Arch.Pharmacol. 1986 PMID: 2936965

Product Documents for Cyanopindolol hemifumarate