Cyclapolin 9

Catalog # Availability Size / Price Qty
3116/10
3116/50
Cat.No. 3116 - Cyclapolin 9 | C9H4F3N3O4S | CAS No. 40533-25-3
1 Image
Description: Selective, ATP-competitive PLK1 inhibitor

Chemical Name: 7-Nitro-5-(trifluoromethyl)-2-benzothiazolecarboxamide-3-oxide

Purity: ≥98%

Product Details
Citations (1)
Reviews

Biological Activity

Selective, ATP-competitive polo-like kinase 1 (PLK1) inhibitor (IC50 = 500 nM).

Technical Data

M.Wt:
307.21
Formula:
C9H4F3N3O4S
Solubility:
Soluble to 25 mM in DMSO and to 10 mM in ethanol
Purity:
≥98%
Storage:
Desiccate at +4°C
CAS No:
40533-25-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Background References

  1. Ligand discovery and virtual screening using the program LIDAEUS.
    Taylor et al.
    Br.J.Pharmacol., 2008;153:S55
  2. Inhibitors of polo-like kinase reveal roles in spindle pole maintenance.
    McInnes et al.
    Nature Chem.Biol., 2006;2:608

Product Datasheets

Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

Citation for Cyclapolin 9

The citations listed below are publications that use Tocris products. Selected citations for Cyclapolin 9 include:

1 Citation: Showing 1 - 1

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

Reviews for Cyclapolin 9

There are currently no reviews for this product. Be the first to review Cyclapolin 9 and earn rewards!

Have you used Cyclapolin 9?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.