Cyprodime hydrochloride

Tocris Bioscience | Catalog # 2601

Selective μ antagonist
Tocris Bioscience

Key Product Details

Description

Selective μ antagonist
View all mu Opioid Receptor Antagonists »

Product Description

Cyprodime hydrochloride is a selective μ-opioid receptor antagonist (Ki values are 5.4, 244.6 and 2187 nM for μ-, δ- and κ-opioid receptors respectively). Reduces levodopa-induced dyskinesia in the MPTP-lesioned primate model of Parkinson's disease.

Product Specifications for Cyprodime hydrochloride

Molecular Weight

391.93

Formula

C22H29NO3.HCl

Storage

Desiccate at +4°C

Purity

≥98% (HPLC)

Chemical Name

17-(Cyclopropylmethyl)-4,14-dimethoxymorphinan-6-one hydrochloride

CAS Number

2387505-50-0

PubChem ID

71628324

InChI Key

MMOBYZBXXHEAAX-NCBCLDNOSA-N

SMILES

O=C3C[C@]24C1=C(OC)C=CC=C1C[C@@H](N(CC5CC5)CC4)[C@@](OC)2CC3.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 39.19 100
Ethanol 39.19 100

Preparing Stock Solutions for Cyprodime hydrochloride

The following data is based on the product molecular weight 391.93.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.55 mL 12.76 mL 25.51 mL
5 mM 0.51 mL 2.55 mL 5.10 mL
10 mM 0.26 mL 1.28 mL 2.55 mL
50 mM 0.05 mL 0.26 mL 0.51 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 10 publications citing the usage of this product.

Product Documents for Cyprodime hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Cyprodime hydrochloride

For research use only

Citations for Cyprodime hydrochloride

Customer Reviews for Cyprodime hydrochloride (1)

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  • Opioid Receptor Antagonist
    Name: Steven Laviolette
    Assay Type: In Vivo
    Verified Customer | Posted 08/22/2018
    Intra-cranial microinfusions for behavioural testing.
    Cyprodime hydrochloride 2601

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