Potent and selective human vasopressin V1B
receptor agonist (Ki
values are 1.2, 151, 240 and 750 nM for V1B
, Oxytocin and V2
receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo
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[1-Deamino-4-cyclohexylalanine] arginine vasopressin: a potent and specific agonist for vasopressin V1b receptors.
Derick et al.
Design of potent and selective agonists for the human vasopressin V1b receptor based on modifications of [deamino-cys1]arginine vasopressin at position 4.
Cheng et al.
Design and synthesis of the frist selective agonists for the rat vasopressin V1b receptor: based on modifications of deamino-[cys1]arginine vasopressin at positions 4 and 8.
Pena et al.
The citations listed below are publications that use Tocris products. Selected citations for d[Cha4]-AVP include:
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