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G-Protein antagonist peptide

1931 2 Citations Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
1931/1
G-Protein antagonist peptide
1 Image
Description: Inhibits G protein activation by GPCRs
Alternative Names: GPAnt-2
Product Details
Citations (2)
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

G-Protein antagonist peptide is a substance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.

Technical Data

M.Wt:
1093.27
Formula:
C57H64N12O9S
Sequence:
XQWFWWM

(Modifications: X = Glp, Trp-3 = Trp-5 = Trp-6 = D-Trp, Met-7 = C-terminal amide)

Solubility:
Soluble to 2 mg/ml in DMSO
Storage:
Desiccate at -20°C
CAS No:
143675-79-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citations for G-Protein antagonist peptide

The citations listed below are publications that use Tocris products. Selected citations for G-Protein antagonist peptide include:

2 Citations: Showing 1 - 2

  1. A Differential Hypofunctionality of Gαi Proteins Occurs in Adolescent Idiopathic Scoliosis and Correlates with the Risk of Disease Progression.
    Authors: Akoume Et al.
    Sci Rep  2019;9:10074
  2. Retromer stops beta-arrestin 1 mediated signaling from internalized cannabinoid 2 receptors.
    Authors: Nogueras-Ortiz
    Mol Biol Cell  2017;28(24):3554

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