G-Protein antagonist peptide
Biological ActivitySubstance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.
(Modifications: X = Glp, Trp-3 = Trp-5 = Trp-6 = D-Trp, Met-7 = C-terminal amide)
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For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding.
Mukai et al.
Citations for G-Protein antagonist peptide
The citations listed below are publications that use Tocris products. Selected citations for G-Protein antagonist peptide include:
2 Citations: Showing 1 - 2
A Differential Hypofunctionality of Gαi Proteins Occurs in Adolescent Idiopathic Scoliosis and Correlates with the Risk of Disease Progression.
Authors: Akoume Et al.
Sci Rep 2019;9:10074
Retromer stops beta-arrestin 1 mediated signaling from internalized cannabinoid 2 receptors.
Mol Biol Cell 2017;28(24):3554
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