GR 125487 sulfamate

  ( 2 citations )    
Product Datasheet
Catalog Number:1658
Chemical Name:5-Fluoro-2-methoxy-[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]-1H-indole-3-methylcarboxylate sulfamate
Product Details
Citations (2)
Supplemental Products
Reviews
Biological Activity
Potent and selective 5-HT4 receptor antagonist (Ki = 0.19 nM for porcine 5-HT4). Centrally active following systemic administration in vivo.
Technical Data
  • M.Wt:
    524.58
  • Formula:
    C19H26FN3O5S.H2NSO3H
  • Solubility:
    Soluble to 10 mM in water with gentle warming
  • Purity:
    >97
  • Storage:
    Desiccate at RT
  • CAS No:
    859502-43-5
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Additional Information
Licensing Caveats:
Sold for research purposes under agreement from GlaxoSmithKline
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for GR 125487 sulfamate include:

2 Citations: Showing 1 - 2
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  1. Astrocytic adenosine receptor A2A and Gs-coupled signaling regulate memory.
    Authors: Orr Et al.
    J Neurosci  2015;18:423
  2. Role of p11 in cellular and behavioral effects of 5-HT4 receptor stimulation.
    Authors: Warner-Schmidt Et al.
    Dis Model Mech  2009;29:1937

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