GSK 2801

Catalog # Availability Size / Price Qty
5635/10
Cat.No. 5635 - GSK 2801 | C20H21NO4S | CAS No. 1619994-68-1
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Description: Selective BAZ2A and BAZ2B inhibitor

Chemical Name: 1-[1-[2-(Methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]ethanone

Purity: ≥98%

Product Details
Reviews

Biological Activity

Selective BAZ2A and BAZ2B inhibitor (IC50 values are 0.40 and 0.43 μM, respectively). Selective for BAZ2A/B over TAF1L and BRD9. Cell permeable and orally available.

External Portal Information

Chemicalprobes.org is a portal that offers independent guidance on the selection and/or application of small molecules for research. The use of GSK2801 is reviewed on the chemical probes website.

Technical Data

M.Wt:
371.45
Formula:
C20H21NO4S
Solubility:
Soluble to 50 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1619994-68-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the GSK 2801 probe summary on the SGC website.

Product Datasheets

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Reconstitution Calculator

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