GSK 2801

Catalog #: 5635 Datasheet / COA / SDS

Discontinued Product

5635 has been discontinued.
View all Bromodomain Inhibitors products.
GSK 2801 | CAS No. 1619994-68-1 | Bromodomain Inhibitors
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Description: Selective BAZ2A and BAZ2B inhibitor

Chemical Name: 1-[1-[2-(Methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]ethanone

Purity: ≥98%

Product Details

Biological Activity

GSK 2801 is a selective BAZ2A and BAZ2B inhibitor (IC50 values are 0.40 and 0.43 μM, respectively). Selective for BAZ2A/B over TAF1L and BRD9. Cell permeable and orally available.

External Portal Information is a portal that offers independent guidance on the selection and/or application of small molecules for research. The use of GSK2801 is reviewed on the chemical probes website.

Technical Data

Soluble to 50 mM in DMSO
Store at -20°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the GSK 2801 probe summary on the SGC website.

Product Datasheets

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