Selective BAZ2A and BAZ2B inhibitor (IC50
values are 0.40 and 0.43 μ
M, respectively). Selective for BAZ2A/B over TAF1L and BRD9. Cell permeable and orally available.
Soluble to 50 mM in DMSO
Store at -20°C
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the GSK 2801 probe summary
on the SGC website.
Discovery and characterization of GSK2801, a selective chemical probe for the bromodomains BAZ2A and BAZ2B.
Chen et al.