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Bromodomain Inhibitors: Products

"Bromodomain Inhibitors" has 53 results in Products.
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(+)-JQ1 

Potent and selective BET bromodomain inhibitor; cell permeable
4499
23 Citations
2 Reviews

MZ 1 

(+)-JQ1 based Degrader (PROTAC®) that preferentially degrades BRD4
6154
8 Citations

dBRD9 

Potent and selective BRD9 Degrader (PROTAC®)
6606
3 Citations

I-BET 151 dihydrochloride 

BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes
4650
7 Citations
2 Reviews

I-BRD9 

Potent and selective BRD9 inhibitor
5591
5 Citations

cis MZ 1 

Negative Control for MZ 1 (Cat. No. 6154)
6155
1 Citation

dBET1 

(+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
6327
1 Citation

dBRD9-A 

Potent BRD9 Degrader (PROTAC®)
6943
1 Citation

dBET6 

Potent and selective (+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
6945

XMD 8-92 

ERK5/BMK1 inhibitor; also BRD4 inhibitor
4132
8 Citations

PFI 1 

BET bromodomain inhibitor
4445
4 Citations

Ischemin sodium salt 

CBP inhibitor; cell permeable
4695

Bromosporine 

Broad spectrum bromodomain inhibitor
4758

SGC-CBP30 

Potent CBP/p300 BRD inhibitor
4889
4 Citations
1 Review

OXF BD 02 

Selective BRD4(1) inhibitor
4928

PFI 3 

Potent and selective SMARCA2/4 and polybromo 1 inhibitor
5072
2 Citations

MS 436 

Potent and selective BRD4(1) inhibitor
5173

BAZ2-ICR 

Selective BAZ2 inhibitor
5266

OF 1 

Selective BRPF1B and BRPF2 inhibitor
5289

CPI 203 

BET bromodomain inhibitor; arrests cell cycle at G1 phase
5331
1 Citation
1 Review

GSK 5959 

Potent and selective BRPF1 inhibitor
5385

NI 57 

Potent and selective BRPF bromodomain inhibitor
5546

PFI 4 

Potent and selective BRPF1B bromodomain inhibitor
5576

BI 9564 

Potent and selective BRD9 and BRD7 inhibitor; orally active
5590
1 Citation

(-)-JQ1 

Negative control for (+)-JQ1
5603
2 Citations

LP 99 

Selective BRD7 and BRD9 inhibitor
5496

ent-LP 99 

Negative Control for LP 99
5497

NVS-CECR2-1 

Potent and selective CECR2 inhibitor
5744

BAY 299 

Potent and selective BRD1 and TAF1 inhibitor
5970

TP 472N 

Negative control for TP 472
5999

TP 472 

Potent BRD9/7 inhibitor
6000
2 Citations

Lin28 1632 

RNA binding protein Lin28 inhibitor; promotes mESC differentiation; also bromodomain inhibitor
6068
3 Citations
1 Review

OTX 015 

BET bromodomain inhibitor; orally bioavailable
6181

GSK 6853 

Potent and selective BRPF1 inhibitor
6198

GSK 9311 hydrochloride 

Negative control for GSK 6853
6203

L Moses dihydrochloride 

High affinity and selective PCAF bromodomain inhibitor
6251
1 Citation

AT 1 

(+)-JQ1 based PROTAC® with selectivity for BRD4
6356
3 Citations
1 Review

I-BET 762 

Potent and high affinity BET bromodomain inhibitor; anti-inflammatory; orally bioavailable.
6521

TP 238 

CECR2 and BPTF/FALZ inhibitor
6670

ZXH 3-26 

Potent and selective BRD4 Degrader (PROTAC®)
6713
1 Citation

VZ 185 

Potent and selective BRD7/9 Degrader (PROTAC®)
6936

cis-VZ 185 

Negative control for VZ 185 (Cat. No. 6936)
6939

CeMMEC1 

TAF1 inhibitor
7139

ARV 771 

Potent BET bromodomain PROTAC®; also degrades BRD-tagged chimeric antigen receptors (CAR) in T cells
7256

SIM1 

Potent and selective trivalent BET Bromodomain Degrader (PROTAC®)
7432

cis-SIM1 

Negative control for SIM1 (Cat. No. 7432)
7433

iBET-BD2 

Potent and selective pan-BD2 inhibitor; orally bioavailable
7458

SGC SMARCA-BRDVIII 

Potent and selective SMARCA2/4 and PB1(bromo 5)-selective SWI/SNF bromodomain inhibitor
7460

NVS MLLT-1 

Selective MLLT1/3 inhibitor
7482

(+)-JQ1 bump, acid functionalized 

Functionalized BET bromodomain ligand; precursor for Tag Degraders
7689
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