NBMPR
Tocris Bioscience | Catalog # 2924
Key Product Details
Description
Product Description
NBMPR is an equilibrative nucleoside transporter 1 (ENT1) inhibitor (Ki values are 0.4 and 2800 nM for hENT1 and hENT2 respectively).
Product Specifications for NBMPR
Molecular Weight
Formula
Storage
Purity
Chemical Name
CAS Number
PubChem ID
InChI Key
SMILES
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 41.94 | 100 |
Preparing Stock Solutions for NBMPR
The following data is based on the product molecular weight 419.41.
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 2.38 mL | 11.92 mL | 23.84 mL |
| 5 mM | 0.48 mL | 2.38 mL | 4.77 mL |
| 10 mM | 0.24 mL | 1.19 mL | 2.38 mL |
| 50 mM | 0.05 mL | 0.24 mL | 0.48 mL |
Calculators
Background References
References are publications that support the biological activity of the product. See our Citations tab to view 19 publications citing the usage of this product.
- Tsujie Human equilibrative nucleoside transporter 1, as a predictor of 5-fluorouracil resistance in human pancreatic cancer. Anticancer Res. 2007 PMID: 17695509
- Lin and Buolamwini Synthesis and flow cytometric evaluation, and identification of highly potent dipyrid. analogues as equilibrative nucleoside transporter 1 inhibitors. J.Med.Chem. 2007 PMID: 17636949
- Ward Kinetic and pharmacological properties of cloned human equilibrative nucleoside transporters, ENT1 and ENT2, stably expressed in nucleoside transporter-deficient PK15 cells. J.Biol.Chem. 2000 PMID: 10722669
Product Documents for NBMPR
Certificate of Analysis
To download a Certificate of Analysis, please enter a lot or batch number in the search box below.
Product Specific Notices for NBMPR
For research use only
Citations for NBMPR
Customer Reviews for NBMPR (1)
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Species: RatAssay Type: In VitroCell Line/Tissue: Primary hippocampal neuronsVerified Customer | Posted 09/26/2025The drug was incubated at 100 nM to specifically inhibit ENT1 function.
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