Modulator of GABAA
receptors. Displays modest selectivity for GABAA
receptors; displays partial agonist activity at α
3- and α
5-containing receptors. Exhibits anxiolytic activity.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Comparative cue generalization profiles of L-838,417, SL651498, zolpidem, CL218,872, ocinaplon, bretazenil, zopiclone, and various benzodiazepines in chlordiazepoxide and zolpidem drug discrimination.
Mirza et al.
Selective anxiolysis produced by ocinaplon, a GABAA receptor modulator.
Lippa et al.
GABAA receptors as targets for novel anxiolytic drugs.
Rupprecht et al.
World J.Biol.Psychiatry, 2006;7:231