GABA-A Receptor Modulators: Products

Subtype-selective GABAA modulator

GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors

Allosteric modulator of GABAA receptors

Potent positive allosteric modulator of GABAA receptors

KV7 channel activator; also GABAA modulator and indirect NMDA antagonist

Ligand of the translocator protein (TSPO); also GABAA receptor potentiator

GluK1 antagonist; inhibits carbonic anhydrase (CA) II and IV; also positive allosteric modulator of GABAA receptors

Postitive allosteric modulator of GABAA receptors

Positive allosteric modulator of GABAA receptors

Positive allosteric modulator of GABAA receptors; displays subunit selectivity

Positive modulator of GABAA receptors; endogenous neurosteroid