GABA-A Receptor Modulators: Products

Subtype-selective GABAA modulator

GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors

Allosteric modulator of GABAA receptors

Potent positive allosteric modulator of GABAA receptors

Antagonist of neurosteroid potentiation and direct gating of GABAA

Positive allosteric modulator of GABAA receptors

Positive allosteric modulator of GABAA receptors; direct agonist at higher concentrations

KV7 channel activator; also GABAA modulator and indirect NMDA antagonist

Ligand of the translocator protein (TSPO); also GABAA receptor potentiator

GluK1 antagonist; inhibits carbonic anhydrase (CA) II and IV; also positive allosteric modulator of GABAA receptors

Postitive allosteric modulator of GABAA receptors

Positive allosteric modulator of GABAA receptors

Positive allosteric modulator of GABAA receptors; displays subunit selectivity

GABAA modulator; anxiolytic

α6β3γ2-selective GABAA positive allosteric modulator

Positive modulator of GABAA receptors; endogenous neurosteroid