2 results for "PPAR gamma/NR1C3" in Products

PPAR gamma/NR1C3 Products

Peroxisome proliferator-activated receptor gamma (PPAR gamma) is a lipid-activated nuclear hormone receptor with roles in adipocyte differentiation, lipid and glucose metabolism, and modulation of immune and inflammatory reactions. PPAR gamma is the receptor for insulin-sensitizing thiazolidinediones, commonly used for the treatment of type 2 diabetes.

Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit

Alternate Names: Gleevec,CGP 57148B
Chemical Name: 4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]benzamide methanesulfonate
Purity: ≥98%
Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit
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EGFR kinase inhibitor. Also estrogen and PPARγ ligand

Chemical Name: 5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one
Purity: ≥98%
EGFR kinase inhibitor. Also estrogen and PPARγ ligand
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