AMG 517

Catalog # Availability Size / Price Qty
5995/10
5995/50

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AMG 517 | CAS No. 659730-32-2 | TRPV Antagonists
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Description: Potent TRPV1 antagonist

Chemical Name: N-[4-[[6-[4-(Trifluoromethyl)phenyl]-4-pyrimidinyl]oxy]-2-benzothiazolyl]acetamide

Purity: ≥98%

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Biological Activity

AMG 517 is a potent TRPV1 antagonist (IC50 = 0.9 nM). Inhibits capsaican-induced flinching and reverses analgesia in an inflammatory pain model in rats. Orally bioavailable.

Technical Data

M.Wt:
430.41
Formula:
C20H13F3N4O2S
Solubility:
Soluble to 10 mM in DMSO
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
659730-32-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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