BCTC

Catalog # Availability Size / Price Qty
3875/10
3875/50
BCTC | CAS No. 393514-24-4 | TRPV Antagonists
1 Image
Description: TRPV1 antagonist

Chemical Name: 4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide

Purity: ≥98%

Product Details
Citations (1)
Supplemental Products
Reviews

Biological Activity

Orally effective vanilloid receptor 1 (TRPV1 receptor) antagonist. Inhibits acid- and capsaicin-induced activation of rat TRPV1 receptors (IC50 values are 6.0 and 35 nM respectively). Displays analgesic properties in rat models of inflammatory and neuropathic pain. CNS penetrant.

Technical Data

M.Wt:
372.89
Formula:
C20H25ClN4O
Solubility:
Soluble to 100 mM in DMSO and to 40 mM in ethanol
Purity:
≥98%
Storage:
Store at RT
CAS No:
393514-24-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

Citation for BCTC

The citations listed below are publications that use Tocris products. Selected citations for BCTC include:

1 Citation: Showing 1 - 1

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

VersaClone cDNA Plasmids

Reviews for BCTC

There are currently no reviews for this product. Be the first to review BCTC and earn rewards!

Have you used BCTC?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.