BCTC

  ( 1 citations )    
Product Datasheet
Catalog Number:3875
Chemical Name:4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide
Product Details
Citations (1)
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Biological Activity
Orally effective vanilloid receptor 1 (TRPV1 receptor) antagonist. Inhibits acid- and capsaicin-induced activation of rat TRPV1 receptors (IC50 values are 6.0 and 35 nM respectively). Displays analgesic properties in rat models of inflammatory and neuropathic pain. CNS penetrant.
Technical Data
  • M.Wt:
    372.89
  • Formula:
    C20H25ClN4O
  • Solubility:
    Soluble to 100 mM in DMSO and to 40 mM in ethanol
  • Purity:
    >98
  • Storage:
    Store at RT
  • CAS No:
    393514-24-4
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Product Datasheets
Citations:

The citations listed below are publications that use Tocris products. Selected citations for BCTC include:

1 Citations: Showing 1 - 1

  1. Elevated expression of transient receptor potential vanilloid type 1 in dorsal root ganglia of rats with endometriosis.
    Authors: Lian Et al.
    Mol Med Rep  2017;16:1920

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