Eplerenone

  ( 1 citations )    
Product Datasheet
Catalog Number:2397
Alternate Names:Inspra, Epoxymexrenone
Chemical Name:(7α,11α,17α)-9,11-Epoxy-17-hydroxy-3-oxo-pregn-4-ene-7,21-dicarboxylic acid γ-lactone methyl ester
Product Details
Citations (1)
Reviews
Biological Activity
Selective mineralocorticoid (aldosterone) receptor antagonist (IC50 = 360 nM). Displays > 27-fold selectivity over androgen, progesterone and estrogen receptors (IC50 > 10 μM). Orally active antihypertensive in vivo.
Technical Data
  • M.Wt:
    414.5
  • Formula:
    C24H30O6
  • Solubility:
    Soluble to 10 mM in DMSO
  • Purity:
    >99
  • Storage:
    Store at RT
  • CAS No:
    107724-20-9
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Product Datasheets
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for Eplerenone include:

1 Citations: Showing 1 - 1

  1. Analysis of insulin sensitivity in adipose tissue of patients with primary aldosteronism.
    Authors: Urbanet Et al.
    Purinergic Signal  2010;95:4037

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