Fananserin

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2645/10
2645/50
Fananserin | CAS No. 127625-29-0 | 5-HT2A Receptor Antagonists
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Description: 5-HT2A antagonist; also D4 antagonist
Alternative Names: RP 62203

Chemical Name: 2-[3-[4-(4-Fluorophenyl)-1-piperazinyl]propyl]-2H-naphthyl[1,8-cd]isothiazole-1,1-dioxide

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Biological Activity

5-HT2A receptor antagonist that also displays high affinity at D4 receptors (Ki values are 0.26, 2.93, 25, 38, 70 and 726 nM for 5-HT2A, D4, H1, α1, 5-HT1A and D2 receptors respectively). Inhibits inositol phosphate formation evoked by 5-HT in vitro (IC50 = 7.76 nM) and antagonizes mescaline-induced head twitches in vivo.

Technical Data

Formula:
C23H24FN3O2S
Solubility:
Soluble to 100 mM in DMSO
Storage:
Store the unopened product at room temperature. Do not use past expiration date.
CAS No:
127625-29-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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