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Catalog Number:4508
Chemical Name:1,2-Dihydro-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-3H-benz[e]indole-3-carboxamide hydrochloride
Product Details
Supplemental Products
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Biological Activity
Inverse agonist of 5-HT2C receptors (pKi = 8.18 at human 5-HT2C INI receptors). Also an antagonist of human α2-adrenoceptors. Displays negligible affinity for α1A-adrenoceptors, histamine H1 receptors and muscarinic M1 receptors.
Inverse agonist of 5-HT2C receptors (pKi = 8.18 at human 5-HT2C INI receptors). Also an antagonist of human α2-adrenoceptors. Displays negligible affinity for α1A-adrenoceptors, histamine H1 receptors and muscarinic M1 receptors.
Technical Data
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M.Wt:452.98
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Formula:C25H28N4O2.HCl
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Solubility:Soluble to 25 mM in water and to 25 mM in DMSO
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Purity:>99
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Storage:Desiccate at RT
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CAS No:847871-78-7
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Product Datasheets
VersaClone cDNA Plasmids
Description
Application
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Human 5-HT2C (NP_000859) VersaClone cDNA
RDC0290
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