SB 221284

Catalog # Availability Size / Price Qty
1379/10
1379/50
5-HT2C Receptor Antagonists Small Molecule
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Description: Potent and selective 5-HT2B and 5-HT2C antagonist

Chemical Name: 2,3-Dihydro-5-(methylthio)-N-3-pyridinyl-6-(trifluoromethyl)-1H-indole-1-carboxamide

Purity: ≥99%

Product Details
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Biological Activity

Potent, selective 5-HT2C/2B receptor antagonist. pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 2B and 2C receptors respectively. Centrally active upon systemic administration in vivo.

Technical Data

M.Wt:
353.36
Formula:
C16H14F3N3OS
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
196965-14-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license

Product Datasheets

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