Chemical Name: (2S)-(+)-5,5-Dimethyl-2-morpholineacetic acid
Biological Activity A selective, competitive and orally active GABAB antagonist. Displays an IC50 of 1.1 μM at GABAB, approximately 60 times that of CGP 35348 (Cat. No. 1245) and no binding affinity for GABAA at concentrations up to 100 μM.
Soluble to 100 mM in water and to 100 mM in phosphate buffered saline
Desiccate at -20°C
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
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