XAC

  ( 5 citations )    
Product Datasheet
Catalog Number:3200
Alternate Names:Xanthine amine congener
Chemical Name:N-(2-Aminoethyl)-2-[4-(2,3,6,7-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]-acetamide dihydrochloride
Product Details
Citations (5)
Supplemental Products
Reviews
Biological Activity
Adenosine receptor antagonist (IC50 values are 1.8 and 114 nM at A1 and A2 receptors respectively). Attenuates adenosine-induced vasodilation and exhibits proconvulsant activity in vivo.
Technical Data
  • M.Wt:
    501.41
  • Formula:
    C21H28N6O4.2HCl
  • Solubility:
    Soluble to 100 mM in DMSO
  • Purity:
    >98
  • Storage:
    Desiccate at RT
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Product Datasheets
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for XAC include:

5 Citations: Showing 1 - 5
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  1. Inverse agonism at the P2Y12 receptor and ENT1 transporter blockade contribute to platelet inhibition by ticagrelor.
    Authors: Aungraheeta Et al.
    Blood  2016;128:2717
  2. Application of BRET to monitor ligand binding to GPCRs.
    Authors: Stoddart Et al.
    Nat Methods  2015;12:661
  3. Caffeine acts through neuronal adenosine A2A receptors to prevent mood and memory dysfunction triggered by chronic stress.
    Authors: Kaster Et al.
    Hepatology  2015;112:7833
  4. Characterization by flow cytometry of fluorescent, selective agonist probes of the A(3) adenosine receptor.
    Authors: Kozma Et al.
    Biochem Pharmacol  2013;85:1171
  5. Regulation of hippocampal cannabinoid CB1 receptor actions by adenosine A1 receptors and chronic caffeine administration: implications for the effects of δ9-tetrahydrocannabinol on spatial memory.
    Authors: Sousa Et al.
    Neuropsychopharmacology  2011;36:472

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VersaClone cDNA Plasmids
Description Application Cat# Citations Images  

Human Adenosine A3 R (NP_065734) VersaClone cDNA

RDC0217
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Human Adenosine A3 R (NP_000668) VersaClone cDNA

RDC0216
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Human Adenosine A2a R (NP_000666) VersaClone cDNA

RDC0214
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Human Adenosine A1 R (NP_000665) VersaClone cDNA

RDC0213
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Mouse Adenosine A1 R (NP_000665) VersaClone cDNA

RDC2041
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Mouse Adenosine A3 R (NP_033761) VersaClone cDNA

RDC0806
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Human Adenosine A2b R (NP_000667) VersaClone cDNA

RDC0215
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Mouse Adenosine A2b R (NP_031439) VersaClone cDNA

RDC2227
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Mouse Adenosine A2a R (NP_033760) VersaClone cDNA

RDC2104
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