8-Cyclopentyl-1,3-dimethylxanthine

Key Product Details

Product Description

8-Cyclopentyl-1,3-dimethylxanthine is a high affinity adenosine A₁ receptor antagonist (pKi = 7.5-8).

Product Specifications for 8-Cyclopentyl-1,3-dimethylxanthine

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for 8-Cyclopentyl-1,3-dimethylxanthine

The following data is based on the product molecular weight 248.28.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	4.03 mL	20.14 mL	40.28 mL
5 mM	0.81 mL	4.03 mL	8.06 mL
10 mM	0.40 mL	2.01 mL	4.03 mL
50 mM	0.08 mL	0.40 mL	0.81 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 9 publications citing the usage of this product.

• Dalpiaz Thermodynamics of full agonist, partial agonist, and antagonist binding to wild-type and mutant adenosine A₁ receptors. Biochem.Pharmacol. 1998 PMID: 9827575

Product Documents for 8-Cyclopentyl-1,3-dimethylxanthine