β-Funaltrexamine hydrochloride

Tocris Bioscience | Catalog # 0926

Irreversible and selective μ antagonist
Tocris Bioscience
Discontinued Product
0926 has been discontinued. View all mu Opioid Receptor Antagonists products.

Key Product Details

Description

Irreversible and selective μ antagonist

Alternative Names

β-FNA
View all mu Opioid Receptor Antagonists »

Product Description

β-Funaltrexamine hydrochloride is a selective μ opioid receptor antagonist.

Licensing Information

Sold with the permission of the University of Minnesota

Product Specifications for β-Funaltrexamine hydrochloride

Molecular Weight

490.99

Formula

C25H30N2O6.HCl

Storage

Store at -20°C

Purity

≥98% (HPLC)

Chemical Name

(E)-4-[[5α,6β)-17-Cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxymorphinan-6-yl]amino]-4-oxo-2-butenoicacid methyl ester hydrochloride

CAS Number

72786-10-8

PubChem ID

44522395

InChI Key

BIPHUOBUKMPSQR-NQGXHZAGSA-N

SMILES

Cl.[H][C@@]12OC3=C4C(C[C@@]5([H])N(CC6CC6)CC[C@@]14[C@@]5(O)CC[C@H]2NC(=O)\C=C\C(=O)OC)=CC=C3O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 9.82 20 with gentle warming
DMSO 49.1 100

Preparing Stock Solutions for β-Funaltrexamine hydrochloride

The following data is based on the product molecular weight 490.99.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.04 mL 10.18 mL 20.37 mL
5 mM 0.41 mL 2.04 mL 4.07 mL
10 mM 0.20 mL 1.02 mL 2.04 mL
50 mM 0.04 mL 0.20 mL 0.41 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 7 publications citing the usage of this product.

Product Documents for β-Funaltrexamine hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for β-Funaltrexamine hydrochloride

For research use only

Citations for β-Funaltrexamine hydrochloride

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