BIM 23042

Name: BIM 23042
Brand: Tocris Bioscience
SKU: 3237

Tocris Bioscience | Catalog # 3237

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Citations (6)

Product Documents

Selective neuromedin B receptor antagonist (NMB-R, BB1)

Discontinued Product

3237 has been discontinued. View all Bombesin Receptor Antagonists products.

Product Description
Product Specifications
Solubility
Calculators
Background References
Product Documents
Specific Notices

Key Product Details

Description

Selective neuromedin B receptor antagonist (NMB-R, BB1)

View all Bombesin Receptor Antagonists »

Product Description

BIM 23042 is a selective neuromedin B receptor (NMB-R, BB₁) antagonist (K_i values are 216 and 18,264 nM for BB₁ and BB₂ receptors respectively). Displays no activity at a range of other receptors.

Product Specifications for BIM 23042

Molecular Weight

1192.46

Formula

C₆₃H₇₃N₁₁O₉S₂

Storage

Desiccate at -20°C

CAS Number

111857-96-6

PubChem ID

16173213

InChI Key

WASLGBPOQJKRMS-AAFDAGAGSA-N

SMILES

[H]N[C@H](CC1=CC2=CC=CC=C2C=C1)C(=O)N[C@H]1CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC1=O)C(C)C)C(=O)N[C@H](CC1=CC2=CC=CC=C2C=C1)C(N)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Soluble to 1mg/ml in 0.1% acetic acid

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 6 publications citing the usage of this product.

Ryan Pharmacological profiles of two bombesin analogues in cells transfected with human neuromedin B receptors. Eur.J.Pharmacol. 1996 PMID: 8813645
Milusheva Role of different bombesin receptor subtypes mediating contractile activity in cat upper gastrointestinal tract. Peptides 1998 PMID: 9533644
Orbuch Discovery of a novel class of neuromedin B receptor antagonists, substituted somatostatin analogues. Mol.Pharmacol. 1993 PMID: 7901752

Product Documents for BIM 23042

Certificate of Analysis

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Product Specific Notices for BIM 23042

For research use only

Citations for BIM 23042

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