CGP 42112

Tocris Bioscience | Catalog # 2569

Selective, high affinity AT2 ligand
Tocris Bioscience

Key Product Details

Description

Selective, high affinity AT2 ligand
View all Additional Angiotensin AT2 Receptor Peptides »

Product Description

CGP 42112 is a selective, high affinity angiotensin AT2 receptor ligand (Ki = 0.24 nM). Displays agonistic properties at proximal tubule AT2 receptors, causes Na+, K+-ATPase inhibition and sodium excretion. Antagonizes Ang-II induced contractions in rabbit aortic rings (IC50 = 1850 nM).

Product Specifications for CGP 42112

Molecular Weight

1052.20

Formula

C52H69N13O11

Storage

Store at -20°C

Purity

≥95% (HPLC)

CAS Number

127060-75-7

PubChem ID

123794

InChI Key

UXGNARZDONUMMK-LRMQDCNJSA-N

SMILES

CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC1=CNC=N1)NC(=O)[C@H](CCCCNC(=O)[C@H](CCCNC(N)=N)NC(=O)OCC1=CC=CC=C1)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)C1=CN=CC=C1)C(O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble to 1mg/ml in water

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 12 publications citing the usage of this product.

Product Documents for CGP 42112

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CGP 42112

For research use only

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